Opioid Receptor Agonist

Opioid Receptor Agonists (171):

Cat. No.	Product Name	Effect	Purity

HY-B0418A

Loperamide hydrochloride	Agonist	99.84%
Loperamide (hydrochloride) (R-18553 (hydrochloride)) is an opioid receptor agonist. Loperamide hydrochloride is a selective and competitive human intestinal carboxylesterases (hiCE) inhibitor. Loperamide hydrochloride has anti-diarrheal effect.

HY-106189

CCI-1008	Agonist
CCI-1008 is an opioid receptor agonist. CCI-1008 can be used for research on nervous system diseases.

HY-12392A

Iprindole hydrochloride	Agonist
Iprindole hydrochloride, an opioid receptor agonist, is a tricyclic antidepressant. Iprindole hydrochloride shortens the immobility time in mice forced swimming test, which can be reversed by the opiate antagonist Naloxone (HY-17417A). Iprindole hydrochloride induces lamellar body formation but devoid of lamellar bodies. Iprindole hydrochloride can be used for the research of depression.

HY-P0183

Nociceptin	Agonist	98.09%
Nociceptin, a heptadecapeptide, is the endogenous ligand of the nociceptin receptor, acting as a potent anti-analgesic.

HY-13716

Noscapine	Agonist	99.98%
Noscapine ((S,R)-Noscapine) is an orally active phthalideisoquinoline alkaloid with potent antitussive. Noscapine exerts its antitussive effects by activating sigma opioid receptors and is a non-competitive Bradykinin inhibitor. Noscapine disrupts microtubule dynamics, induces mitotic arrest and apoptosis. Noscapine possesses anticancer, neuroprotective, anti-inflammatory activities, and can cross the blood-brain barrier.

HY-105343

BW-180C	Agonist	99.92%
BW-180C ([D-Ala2, D-Leu5]-Enkephalin; DADLE) is an δ opioid receptor (DOR) agonist, which belongs to the enkephalin family. Neuroprotective agent. BW-180C reversibly inhibits cellular transcription in neurons without causing cell injury.

HY-P0179

β-Casomorphin, bovine	Agonist	99.89%
β-Casomorphin, bovine (β-Casomorphin-7 (bovine) ) is a opioid peptide with an IC₅₀ of 14 μM in an Opioid receptors binding assay.

HY-13101

MCOPPB trihydrochloride	Agonist	99.98%
MCOPPB trihydrochloride is a nociceptin receptor agonist with pKi of 10.

HY-15997B

(±)-U-50488 hydrochloride	Agonist	99.73%
(±)-U-50488 ((±)-Trans-(1R,2R)-U-50488) hydrochloride is a selective κ opioid receptor (KOR) agonist.

HY-B0418AR

Loperamide hydrochloride (Standard)	Agonist
Loperamide (hydrochloride) (Standard) is the analytical standard of Loperamide (hydrochloride). This product is intended for research and analytical applications. Loperamide (hydrochloride) (R-18553 (hydrochloride)) is an opioid receptor agonist. Loperamide hydrochloride is a selective and competitive human intestinal carboxylesterases (hiCE) inhibitor. Loperamide hydrochloride has anti-diarrheal effect.

HY-P1337

Dynorphin B (1-13)	Agonist	98.49%
Dynorphin B (1-13) acts as an agonist on opioid κ-receptor.

HY-P3870A

DALDA acetate	Agonist	99.78%
DALDA acetate is a potent and highly selective μ-opioid receptor agonist with a K_i of 1.69 nM. DALDA acetate shows antinociceptive and respiratory effects.

HY-13716A

Noscapine hydrochloride	Agonist	99.87%
Noscapine ((S,R)-Noscapine) hydrochloride is an orally active phthalideisoquinoline alkaloid with potent antitussive. Noscapine hydrochloride exerts its antitussive effects by activating sigma opioid receptors and is a non-competitive Bradykinin inhibitor. Noscapine hydrochloride disrupts microtubule dynamics, induces mitotic arrest and apoptosis. Noscapine hydrochloride possesses anticancer, neuroprotective, anti-inflammatory activities, and can crosse the blood-brain barrier.

HY-P3609

CR 665	Agonist	99.66%
CR 665 (JNJ 38488502) is a peripherally selective κ-opioid agonist. CR 665 can activate the kappa opioid receptor with EC₅₀ value of 10.9 nM. CR 665 can be used for the research of peripheral pain.

HY-107722

SCH 221510	Agonist	99.06%
SCH 221510 is a potent, orally active and selective NOP (nociceptin opioid receptor) agonist, with an EC₅₀ of 12 nM and K_i of 0.3 nM. SCH 221510 shows an anxiolytic-like effect.

HY-P1470

[Leu5]-Enkephalin, amide	Agonist	99.76%
[Leu5]-Enkephalin, amide is a δ opioid receptor agonist.

HY-P3445A

Anrikefon acetate	Agonist	99.68%
Anrikefon (HSK21542) acetate is a kappa opioid receptor agonist with analgesic effect.

HY-107747

GR 89696	Agonist	99.88%
GR 89696 is a highly selective κ2 opioid receptor agonist with potential to prevent pruritus.

HY-P1302

Orphanin FQ(1-11)	Agonist	99.83%
Orphanin FQ(1-11), a orphanin FQ or nociceptin (OFQ/N) fragment, is a potent NOP receptor (ORL-1; OP4) agonist, with a K_i of 55 nM. Orphanin FQ(1-11) has no affinity for μ, δ, κ1 and κ3 receptors (K_i>1000 nM). Orphanin FQ(1-11) is analgesic in CD-1 mice.

HY-14157

ADL-5747	Agonist	99.82%
ADL-5747 is a selective and orally active agonist of the δ-opioid receptor (DOR). By binding to the δ-opioid receptors, ADL-5747 activates these receptors, thereby playing a role in pain management pathways. ADL-5747 can be used for research into pain management mechanisms.

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